S. Yu. Vostruhina, A. N. Reznikov, Yu. N. Klimochkin
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引用次数: 0
Abstract
3-Phosphorylmethyl-3-R-indolin-2-ones were synthesized by the cascade Heck cyclization—phosphorylation of N-(2-iodophenyl)acrylamides and hydrophosphoryl compounds. In the presence of the PdCl2/(S)-Monophos catalytic system, a racemic product was obtained; while, the (R,R)-DIOP ligand provided small chiral induction (up to 15% ee).
期刊介绍：
Publishing nearly 500 original articles a year, by leading Scientists from Russia and throughout the world, Russian Chemical Bulletin is a prominent international journal. The coverage of the journal spans practically all areas of fundamental chemical research and is presented in five sections:
General and Inorganic Chemistry;
Physical Chemistry;
Organic Chemistry;
Organometallic Chemistry;
Chemistry of Natural Compounds and Bioorganic Chemistry.
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