Anastasiia A Uspenskaia, Irina A Doroshenko, Kseniia A Popovicheva, Nazar V Shmychkov, Ekaterina V Pryakhina, Radik R Shafikov, Dmitrii A Skvortsov, Mikhail K Beklemishev, Olga V Zaborova, Tatiana A Podrugina, Aleksei E Machulkin, Elena K Beloglazkina
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引用次数: 0
Abstract
We report a modified carbocyanine-based asymmetric fluorescent dye, suitable for the azide-alkyne cycloaddition reaction, that possesses promising photochemical properties (Φfl = 0,49). As an example of usage of the new fluorophore, it was conjugated to a ligand targeting prostate-specific membrane antigen (PSMA), one of the widely utilized prostate cancer markers.
期刊介绍：
Bioorganic & Medicinal Chemistry Letters presents preliminary experimental or theoretical research results of outstanding significance and timeliness on all aspects of science at the interface of chemistry and biology and on major advances in drug design and development. The journal publishes articles in the form of communications reporting experimental or theoretical results of special interest, and strives to provide maximum dissemination to a large, international audience.
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