Xianhe Fang , Jiaxing Lv , Shuxin Yang , Mingyu Ma , Runzhe Yang , Yi Bi
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引用次数: 0
Abstract
Herein, we describe a cascade C(sp3)-H bond functionalization/cyclization reaction for the synthesis of 3,3-disubstituted oxindoles. The reaction is catalyzed by decatungstate anion under near-ultraviolet light irradiation. Functionalization of aliphatic C(sp3)−H bonds occurs efficiently through this catalytic reaction. Furthermore, the selected products exhibited inhibitory effects on LPS-induced macrophage nitric oxide release.
期刊介绍：
Tetrahedron publishes full accounts of research having outstanding significance in the broad field of organic chemistry and its related disciplines, such as organic materials and bio-organic chemistry.
Regular papers in Tetrahedron are expected to represent detailed accounts of an original study having substantially greater scope and details than that found in a communication, as published in Tetrahedron Letters.
Tetrahedron also publishes thematic collections of papers as special issues and ''Reports'', commissioned in-depth reviews providing a comprehensive overview of a research area.
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