Targeted Complexes of Lanthanide(III) Ions as Therapeutic and Diagnostic Pharmaceuticals

Mark Woods , Zoltan Kovacs , A.Dean Sherry
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镧系(III)离子靶向配合物作为治疗和诊断药物
镧系离子的物理、磁性和核特性使其成为诊断和治疗药物的理想用途。生物技术的最新创新为此类药物的设计开辟了新的可能性。通过将合适的靶向载体与金属螯合物偶联,可以靶向组织类型、细胞类型、单个蛋白质甚至特定核酸序列。这篇综述介绍了这些配合物靶向的最新进展,并讨论了它们在开发新型无机药物中的潜力。
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