基于片段的筛选方法揭示了寻找tau-tubulin激酶1异位抑制剂的非正位口袋

Robert P. Hayes, Edward DiNunzio, Mahdieh Yazdani, Justyna Sikorska, Yili Chen, S. Tyagarajan, Younghee Park, Amy Lee, Cesar Reyes, Daniel Burschowsky, Matthias Zebisch, Yangsi Ou, Marina Bukhtiyarova, Shahriar Niroomand, Yuan Tian, Shawn J. Stachel, Hua Su, Jacqueline D. Hicks, Daniel F. Wyss
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Fragment-based screening approach reveals non-orthosteric pockets in the search for allosteric inhibitors of tau-tubulin kinase 1
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