Samir, MESSAOUDI, Sokna , Bazzi, Ameni , Hadj Mohamed, Dmytro , Ryzhakov, Juba , Ghouilem, Mehdi A. , Beniddir, Vincent , Gandon
{"title":"非对映选择性 C(sp3)-H-环化实现新一代环烷糖肽的设计","authors":"Samir, MESSAOUDI, Sokna , Bazzi, Ameni , Hadj Mohamed, Dmytro , Ryzhakov, Juba , Ghouilem, Mehdi A. , Beniddir, Vincent , Gandon","doi":"10.26434/chemrxiv-2024-zgxwt","DOIUrl":null,"url":null,"abstract":"Here we report a macrocyclization route towards the\nsynthesis of glycophane peptides by a selective C-H arylation of the anomeric bond. This approach demonstrates the power of Pd-catalysis\nC-H activation to access unfamiliar cyclic peptides","PeriodicalId":9813,"journal":{"name":"ChemRxiv","volume":null,"pages":null},"PeriodicalIF":0.0000,"publicationDate":"2024-09-13","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":"0","resultStr":"{\"title\":\"Diastereoselective Anomeric C(sp3)-H Cyclization Towards the Design of New Generations of Cyclophane-Braced Glycopeptides\",\"authors\":\"Samir, MESSAOUDI, Sokna , Bazzi, Ameni , Hadj Mohamed, Dmytro , Ryzhakov, Juba , Ghouilem, Mehdi A. , Beniddir, Vincent , Gandon\",\"doi\":\"10.26434/chemrxiv-2024-zgxwt\",\"DOIUrl\":null,\"url\":null,\"abstract\":\"Here we report a macrocyclization route towards the\\nsynthesis of glycophane peptides by a selective C-H arylation of the anomeric bond. This approach demonstrates the power of Pd-catalysis\\nC-H activation to access unfamiliar cyclic peptides\",\"PeriodicalId\":9813,\"journal\":{\"name\":\"ChemRxiv\",\"volume\":null,\"pages\":null},\"PeriodicalIF\":0.0000,\"publicationDate\":\"2024-09-13\",\"publicationTypes\":\"Journal Article\",\"fieldsOfStudy\":null,\"isOpenAccess\":false,\"openAccessPdf\":\"\",\"citationCount\":\"0\",\"resultStr\":null,\"platform\":\"Semanticscholar\",\"paperid\":null,\"PeriodicalName\":\"ChemRxiv\",\"FirstCategoryId\":\"1085\",\"ListUrlMain\":\"https://doi.org/10.26434/chemrxiv-2024-zgxwt\",\"RegionNum\":0,\"RegionCategory\":null,\"ArticlePicture\":[],\"TitleCN\":null,\"AbstractTextCN\":null,\"PMCID\":null,\"EPubDate\":\"\",\"PubModel\":\"\",\"JCR\":\"\",\"JCRName\":\"\",\"Score\":null,\"Total\":0}","platform":"Semanticscholar","paperid":null,"PeriodicalName":"ChemRxiv","FirstCategoryId":"1085","ListUrlMain":"https://doi.org/10.26434/chemrxiv-2024-zgxwt","RegionNum":0,"RegionCategory":null,"ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":null,"EPubDate":"","PubModel":"","JCR":"","JCRName":"","Score":null,"Total":0}
Diastereoselective Anomeric C(sp3)-H Cyclization Towards the Design of New Generations of Cyclophane-Braced Glycopeptides
Here we report a macrocyclization route towards the
synthesis of glycophane peptides by a selective C-H arylation of the anomeric bond. This approach demonstrates the power of Pd-catalysis
C-H activation to access unfamiliar cyclic peptides
京公网安备 11010802042870号
京ICP备2023020795号-1
分享
求助内容：
应助结果提醒方式：
扫码关注我们
