Selectfluor从吲哚-2- 1中提取3-氟辛孔

IF 2.2 3区化学 Q2 CHEMISTRY, ORGANIC Tetrahedron Pub Date : 2025-06-01 Epub Date: 2025-02-26 DOI:10.1016/j.tet.2025.134556

Hui Qin , Guo-Liang Wei , Fu-Wei Wang , Xiao-Hong Mao , Mei-Hua Bao , Yi-Wen Zhang , Ping Huang , Xiao-Wei Zheng

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引用次数: 0

摘要

本文利用选择性氟作为一种经济高效的氟化试剂，提出了一种在温和条件下对多种吲哚-2- 1进行氟化的方法。值得注意的是，该议定书是在环境友好的条件下进行的，有助于以中等至较高的产量将各种取代的吲哚-2- 1生成相应的氟化吲哚-2- 1，所有这些都不需要碱源或加热。

本文章由计算机程序翻译，如有差异，请以英文原文为准。

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3-Fluorooxindoles from indolin-2-ones by Selectfluor

Herein, a practical and efficient method for fluorinating various indolin-2-ones under mild conditions was presented, utilizing selectfluor as a cost-effective fluorination reagent. Notably, the protocol operated under environmentally friendly conditions, facilitating the generation of various substituted indolin-2-ones into corresponding fluorinated indolin-2-ones in moderate to good yields, all without the need for an alkali source or heating.

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来源期刊

Tetrahedron 化学-有机化学

CiteScore

3.90

自引率

4.80%

发文量

439

审稿时长

34 days

期刊介绍： Tetrahedron publishes full accounts of research having outstanding significance in the broad field of organic chemistry and its related disciplines, such as organic materials and bio-organic chemistry. Regular papers in Tetrahedron are expected to represent detailed accounts of an original study having substantially greater scope and details than that found in a communication, as published in Tetrahedron Letters. Tetrahedron also publishes thematic collections of papers as special issues and ''Reports'', commissioned in-depth reviews providing a comprehensive overview of a research area.