Pavel Golubev, Olga Bakulina, Dmitry Dar'in, Mikhail Krasavin
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ChemInform Abstract: Indoline-Based Constrained Peptidomimetic Motifs Obtained via the Joullie—Ugi Reaction of Indolenines.
Sterically demanding indolenines are employed as cyclic imine substrates in the title reaction with isocyanides and carboxylic acids, resulting in a new type of conformationally constrained indoline-based peptidomimetics.