Mathilde A. C. H. Janssen, Rico Rappard, Tom Dekker, Mitchel Heiming, Marjolijn Beens, Dyon Pieters, Brian H. M. Kuijpers, Jorg C. J. Benningshof, Maikel Wijtmans, Iwan J. P. de Esch, Daniel Blanco-Ania, Floris P. J. T. Rutjes
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引用次数: 0
Abstract
Cyclobutanes have attracted significant interest in medicinal chemistry because of their unique structure and potential advantages in pharmacological properties. In this study a two-diversification-point library of cyclobutanesulfonamides with either carbamates or triazoles was synthesized through a hyperbaric [2+2] cycloaddition reaction between ethenesulfonyl fluoride and tert-butyl vinyl ether as the key step.
期刊介绍：
The European Journal of Organic Chemistry (2019 ISI Impact Factor 2.889) publishes Full Papers, Communications, and Minireviews from the entire spectrum of synthetic organic, bioorganic and physical-organic chemistry. It is published on behalf of Chemistry Europe, an association of 16 European chemical societies.
The following journals have been merged to form two leading journals, the European Journal of Organic Chemistry and the European Journal of Inorganic Chemistry:
Liebigs Annalen
Bulletin des Sociétés Chimiques Belges
Bulletin de la Société Chimique de France
Gazzetta Chimica Italiana
Recueil des Travaux Chimiques des Pays-Bas
Anales de Química
Chimika Chronika
Revista Portuguesa de Química
ACH—Models in Chemistry
Polish Journal of Chemistry.
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