Yaqi Zhang, Qiang Ni, Rihui Cao, Long Jiang, Liqin Qiu
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引用次数: 0
Abstract
A stereoselective Ni−Al bimetal-catalyzed C−H alkenylation of quinazolinones with alkynes has been successfully developed. Good selectivity of Z-type quinazolinone products was obtained using readily available substrates, which exhibits a trans-configuration opposite to the conventional alkynylation reactions and improves the diversity of quinazolinone compounds. In addition, the reaction process was further explored through KIE and other control experiments, and a possible mechanism was proposed.
期刊介绍：
The European Journal of Organic Chemistry (2019 ISI Impact Factor 2.889) publishes Full Papers, Communications, and Minireviews from the entire spectrum of synthetic organic, bioorganic and physical-organic chemistry. It is published on behalf of Chemistry Europe, an association of 16 European chemical societies.
The following journals have been merged to form two leading journals, the European Journal of Organic Chemistry and the European Journal of Inorganic Chemistry:
Liebigs Annalen
Bulletin des Sociétés Chimiques Belges
Bulletin de la Société Chimique de France
Gazzetta Chimica Italiana
Recueil des Travaux Chimiques des Pays-Bas
Anales de Química
Chimika Chronika
Revista Portuguesa de Química
ACH—Models in Chemistry
Polish Journal of Chemistry.
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