Toward a broad-based antisense technology.

R W Wagner
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Detection of ribonuclease H-generated mRNA fragments in human leukemia cells following reversible membrane permeabilization in the presence of antisense oligodeoxynucleotides. (2'-5')-Oligo-3'-deoxynucleotides: selective binding to single-stranded RNA but not DNA. Inhibition of protein-tyrosine kinase activity in intact cells by the aptameric action of oligodeoxynucleotides. Helix-stabilizing compounds CC-1065 and U-71,184 bind to RNA-DNA and DNA-DNA duplexes containing modified internucleotide linkages and stabilize duplexes against thermal melting. Toward a broad-based antisense technology.
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