Changkuo Zhao , Linming Zuo , Xi Ke , Xianheng Wang
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A simple method for Michael addition at C-5 of Camptothecin has been developed to construct 5-CPT derivatives. The addition products were obtained with moderate yields, and the structures of the target compounds were characterized by 1H NMR, 13C NMR, and HRMS spectra. The feasibility of various Michael addition acceptors for this reaction has also been investigated.
期刊介绍：
Journal of Saudi Chemical Society is an English language, peer-reviewed scholarly publication in the area of chemistry. Journal of Saudi Chemical Society publishes original papers, reviews and short reports on, but not limited to:
•Inorganic chemistry
•Physical chemistry
•Organic chemistry
•Analytical chemistry
Journal of Saudi Chemical Society is the official publication of the Saudi Chemical Society and is published by King Saud University in collaboration with Elsevier and is edited by an international group of eminent researchers.
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