Alexander N. Larin, Anastasia A. Borovleva, Oleg P. Demidov, Elena K. Avakyan, Alexander A. Zubenko, Diana Yu. Pobedinskaya, Artem P. Ermolenko, Stepan E. Kolosov, Ivan V. Borovlev
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Selective SNH Alkylamination of 3(5,6,7,8)-Nitroquinoline and 5-Nitroisoquinoline in an Aqueous Medium
Direct oxidative SNH alkylamination of 3-, 5-, 6-, 7-, 8-nitroquinolines and 5-nitroisoquinoline in an aqueous solution of an aliphatic amines gives rise to the corresponding alkylamino and dialkylamino derivatives of these nitrohetarenes. The nitro group solely dictates the regioselectivity of reactions. The antibacterial activity of some of them has been studied.
期刊介绍：
Organic chemistry is the fundamental science that stands at the heart of chemistry, biology, and materials science. Research in these areas is vigorous and truly international, with three major regions making almost equal contributions: America, Europe and Asia. Asia now has its own top international organic chemistry journal—the Asian Journal of Organic Chemistry (AsianJOC)
The AsianJOC is designed to be a top-ranked international research journal and publishes primary research as well as critical secondary information from authors across the world. The journal covers organic chemistry in its entirety. Authors and readers come from academia, the chemical industry, and government laboratories.
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