Zizhen Liu, Zhiguang Zhai, Daoshun Wu, Jianhe Wei, Zhen Yang, Prof. Dr. Jie Zhang, Prof. Dr. Lei Wang
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引用次数: 0
Abstract
A Brønsted acid catalyzed direct and dual C−H amination of carbazoles and indolocarbazoles with N-Ts iminoquinone acetal is reported. It is characterized that the mentioned C−H amination was determined by the selection of catalysts and the molar ratio of the starting materials. The efficiency of this protocol was showcased by diverse carbazolylamine and indolocarbazolylamine assemblies. The late-stage functionalization of a series of natural products fully illustrates the synthetic value of this methodology.
期刊介绍：
Organic chemistry is the fundamental science that stands at the heart of chemistry, biology, and materials science. Research in these areas is vigorous and truly international, with three major regions making almost equal contributions: America, Europe and Asia. Asia now has its own top international organic chemistry journal—the Asian Journal of Organic Chemistry (AsianJOC)
The AsianJOC is designed to be a top-ranked international research journal and publishes primary research as well as critical secondary information from authors across the world. The journal covers organic chemistry in its entirety. Authors and readers come from academia, the chemical industry, and government laboratories.
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