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Novel Peripherally Selective Cannabinoid Receptor 1 Neutral Antagonist Improves Metabolic Dysfunction-Associated Steatotic Liver Disease in Mice 新型外周选择性大麻素受体 1 中性拮抗剂可改善小鼠代谢功能障碍相关性脂肪肝病症
Pub Date : 2024-08-08 DOI: 10.1021/acsptsci.4c00356
Lucas T. Laudermilk, J. Schlosburg, Elaine A. Gay, Ann M. Decker, Aaron Williams, Rubica Runton, Vineetha Vasukuttan, Archana Kotiya, G. Amato, Rangan Maitra
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引用次数: 0
Targeting Matrix Metalloproteinase-9 for Therapeutic Intervention in Diabetic Foot Ulcers 靶向基质金属蛋白酶-9 治疗糖尿病足溃疡
Pub Date : 2024-07-16 DOI: 10.1021/acsptsci.4c00263
Mayland Chang
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引用次数: 0
Exploring an Intracellular Allosteric Site of CC-Chemokine Receptor 4 from 3D Models, Probe Simulations, and Mutagenesis 从三维模型、探针模拟和突变中探索 CC-Chemokine Receptor 4 的细胞内异构位点
Pub Date : 2024-07-16 DOI: 10.1021/acsptsci.4c00330
Tianyi Ding, Abdul-Akim Guseinov, Graeme Milligan, Bianca Plouffe, Irina G. Tikhonova
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引用次数: 0
Rapid-Test Kit for Cardiac Troponin I: A Reliable Enzyme-Linked-Immuno-Substrate-Assay-Based Biosensor for Daily-Use Naked-Eye Detection and Pharmacokinetic Studies for Myocardial Infarction in Cardiovascular Disease 心肌肌钙蛋白 I 快速检测试剂盒:基于酶联免疫底物分析的可靠生物传感器,用于心血管疾病中心肌梗死的日用裸眼检测和药代动力学研究
Pub Date : 2024-07-15 DOI: 10.1021/acsptsci.4c00218
Yu-Fang Hsieh, Kuan-Jiuh Lin
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引用次数: 0
A First Insight into the Developability of an Immunoglobulin G3: A Combined Computational and Experimental Approach 首次洞察免疫球蛋白 G3 的可开发性:计算与实验相结合的方法
Pub Date : 2024-07-15 DOI: 10.1021/acsptsci.4c00271
Georgina B. Armstrong, Alan Lewis, Vidhi Shah, Paul Taylor, Craig Jamieson, Glenn A. Burley, William Lewis, Zahra Rattray
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引用次数: 0
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ACS Pharmacology & Translational Science
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