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ASPET 2023 Annual Meeting Abstract - Cellular and Molecular Pharmacology最新文献

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Investigating the Intertwine Effect of Insulin Resistance and Lipocalin Prostaglandin D2 Synthase in Non-alcoholic Fatty Liver Disease using HepG2 Cells 利用HepG2细胞研究非酒精性脂肪肝患者胰岛素抵抗和脂钙素前列腺素D2合成酶的相互作用
Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.539140
Rhema Khairnar, Md Asrarul Islam, Sunil Kumar
Abstract
摘要
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引用次数: 0
Molecular regulation of G protein prenylation under sub-optimal conditions 次优条件下G蛋白戊酰化的分子调控
Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.558790
A. Karunarathne, M. Tennakoon, Waruna Thotamune, John L. Payton
{"title":"Molecular regulation of G protein prenylation under sub-optimal conditions","authors":"A. Karunarathne, M. Tennakoon, Waruna Thotamune, John L. Payton","doi":"10.1124/jpet.122.558790","DOIUrl":"https://doi.org/10.1124/jpet.122.558790","url":null,"abstract":"","PeriodicalId":406842,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Cellular and Molecular Pharmacology","volume":"38 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"114946196","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Spatial Compartmentalization of mTORC1 to the Nucleus to Regulate Transcription and Impact Nuclear Erk Signaling mTORC1到细胞核的空间区隔调节转录和影响核Erk信号传导
Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.169530
A. Şahan, Yanghao Zhong, C. Sauceda, D. Gonzalez, Jin Zhang
{"title":"Spatial Compartmentalization of mTORC1 to the Nucleus to Regulate Transcription and Impact Nuclear Erk Signaling","authors":"A. Şahan, Yanghao Zhong, C. Sauceda, D. Gonzalez, Jin Zhang","doi":"10.1124/jpet.122.169530","DOIUrl":"https://doi.org/10.1124/jpet.122.169530","url":null,"abstract":"","PeriodicalId":406842,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Cellular and Molecular Pharmacology","volume":"75 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"131786314","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Zyflamend, a novel approach for the treatment of acute pancreatitis Zyflamend,治疗急性胰腺炎的新方法
Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.229630
Ahmed Elshaarrawi, Ahmed Bettaieb, Presley D Dowker-Key
{"title":"Zyflamend, a novel approach for the treatment of acute pancreatitis","authors":"Ahmed Elshaarrawi, Ahmed Bettaieb, Presley D Dowker-Key","doi":"10.1124/jpet.122.229630","DOIUrl":"https://doi.org/10.1124/jpet.122.229630","url":null,"abstract":"","PeriodicalId":406842,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Cellular and Molecular Pharmacology","volume":"232 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"134590815","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Without a Trace: The Pirin and NF-κB Interaction 无迹可循:Pirin与NF-κB的相互作用
Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.264930
Melissa Meschkewitz, E. Lisabeth, R. Neubig
Abstract
摘要
{"title":"Without a Trace: The Pirin and NF-κB Interaction","authors":"Melissa Meschkewitz, E. Lisabeth, R. Neubig","doi":"10.1124/jpet.122.264930","DOIUrl":"https://doi.org/10.1124/jpet.122.264930","url":null,"abstract":"Abstract","PeriodicalId":406842,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Cellular and Molecular Pharmacology","volume":"25 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"121698090","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Insurmountable Antagonism by Buprenorphine at Human Mu Opioid Receptors 丁丙诺啡对人Mu阿片受体的不可克服拮抗作用
Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.168480
M. Wedemeyer, K. Berg, W. Clarke
{"title":"Insurmountable Antagonism by Buprenorphine at Human Mu Opioid Receptors","authors":"M. Wedemeyer, K. Berg, W. Clarke","doi":"10.1124/jpet.122.168480","DOIUrl":"https://doi.org/10.1124/jpet.122.168480","url":null,"abstract":"","PeriodicalId":406842,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Cellular and Molecular Pharmacology","volume":"11 1 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"125814435","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Molecular Dynamics Studies for Nirmatrelvir and the Main Protease from Variants of the Severe Acute Respiratory Syndrome Coronavirus-2 (SARS-CoV-2) 严重急性呼吸综合征冠状病毒-2 (SARS-CoV-2)变异体对Nirmatrelvir及其主要蛋白酶的分子动力学研究
Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.196270
K. Frey, Ongshu Dutta, Lilian Tran, Brandon Yin, Andrew Makarus, Raymond Marmol, Youssef Dawood
{"title":"Molecular Dynamics Studies for Nirmatrelvir and the Main Protease from Variants of the Severe Acute Respiratory Syndrome Coronavirus-2 (SARS-CoV-2)","authors":"K. Frey, Ongshu Dutta, Lilian Tran, Brandon Yin, Andrew Makarus, Raymond Marmol, Youssef Dawood","doi":"10.1124/jpet.122.196270","DOIUrl":"https://doi.org/10.1124/jpet.122.196270","url":null,"abstract":"","PeriodicalId":406842,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Cellular and Molecular Pharmacology","volume":"4 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"130488225","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Subcellular Localization Analysis of Sigma 1 Receptor (S1R) and Binding Immunoglobulin Protein (BiP) for Identification of Antagonists versus Agonists Sigma 1受体(S1R)和结合免疫球蛋白蛋白(BiP)的亚细胞定位分析用于鉴别拮抗剂和激动剂
Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.176040
F. Simin, Joseph M. Schober
Abstract
摘要
{"title":"Subcellular Localization Analysis of Sigma 1 Receptor (S1R) and Binding Immunoglobulin Protein (BiP) for Identification of Antagonists versus Agonists","authors":"F. Simin, Joseph M. Schober","doi":"10.1124/jpet.122.176040","DOIUrl":"https://doi.org/10.1124/jpet.122.176040","url":null,"abstract":"Abstract","PeriodicalId":406842,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Cellular and Molecular Pharmacology","volume":"10 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"123979194","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Identification of a sequence of the activity-dependent neuroprotective protein (ADNP) that is necessary for its interaction with G??i1 活性依赖性神经保护蛋白(ADNP)序列的鉴定是其与G??i1
Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.162450
N. Momplaisir, N. Chandan, A. Smrcka
{"title":"Identification of a sequence of the activity-dependent neuroprotective protein (ADNP) that is necessary for its interaction with G??i1","authors":"N. Momplaisir, N. Chandan, A. Smrcka","doi":"10.1124/jpet.122.162450","DOIUrl":"https://doi.org/10.1124/jpet.122.162450","url":null,"abstract":"","PeriodicalId":406842,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Cellular and Molecular Pharmacology","volume":"31 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"131633869","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Role of orphan G Protein-Coupled Receptor GPRC5B in retinoic acid induced depressive-like behaviors 孤儿G蛋白偶联受体GPRC5B在维甲酸诱导的抑郁样行为中的作用
Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.155670
Wenqi Fu, L. Franchini, C. Orlandi, N. Wettschureck
{"title":"Role of orphan G Protein-Coupled Receptor GPRC5B in retinoic acid induced depressive-like behaviors","authors":"Wenqi Fu, L. Franchini, C. Orlandi, N. Wettschureck","doi":"10.1124/jpet.122.155670","DOIUrl":"https://doi.org/10.1124/jpet.122.155670","url":null,"abstract":"","PeriodicalId":406842,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Cellular and Molecular Pharmacology","volume":"14 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"116906232","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
期刊
ASPET 2023 Annual Meeting Abstract - Cellular and Molecular Pharmacology
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