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Progress in medicinal chemistry最新文献

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The discovery of raltegravir, an integrase inhibitor for the treatment of HIV infection. 发现用于治疗HIV感染的整合酶抑制剂雷替格拉韦。
Q1 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2008-01-01 DOI: 10.1016/S0079-6468(07)00001-X
Michael Rowley
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引用次数: 50
Histone deacetylase inhibitors: a novel class of anti-cancer agents on its way to the market. 组蛋白去乙酰化酶抑制剂:一类即将上市的新型抗癌药物。
Q1 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2008-01-01 DOI: 10.1016/S0079-6468(07)00005-7
Matthias Körner, Ulrich Tibes
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引用次数: 12
5-HT2C ligands: recent progress. 5-HT2C配体:最新进展。
Q1 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2008-01-01 DOI: 10.1016/S0079-6468(07)00006-9
Nathaniel J T Monck, Guy A Kennett
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引用次数: 25
Hit and Lead identification: efficient practices for drug discovery. Hit和Lead鉴定:药物发现的有效实践。
Q1 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2007-01-01 DOI: 10.1016/S0079-6468(06)45501-6
Robert A Goodnow, Paul Gillespie
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引用次数: 17
Tuberculosis chemotherapy: recent developments and future perspectives. 结核病化疗:最近的发展和未来的展望。
Q1 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2007-01-01 DOI: 10.1016/S0079-6468(06)45504-1
Veemal Bhowruth, Lynn G Dover, Gurdyal S Besra
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引用次数: 34
DPPIV inhibition: promising therapy for the treatment of type 2 diabetes. DPPIV抑制:治疗2型糖尿病的有希望的疗法。
Q1 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2007-01-01 DOI: 10.1016/S0079-6468(06)45502-8
Paul E Wiedeman
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引用次数: 23
Recent progress toward nonpeptide ligands for the melanocortin-4 receptor. 黑素皮质素-4受体非肽配体研究进展。
Q1 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2007-01-01 DOI: 10.1016/S0079-6468(06)45503-X
Chen Chen
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引用次数: 12
Blunting the Swiss army knife of hepatitis C virus: inhibitors of NS3/4A protease. 钝化丙型肝炎病毒的瑞士军刀:NS3/4A蛋白酶抑制剂。
Q1 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2006-01-01 DOI: 10.1016/S0079-6468(05)44402-1
Peter W White, Montse Llinas-Brunet, Michael Bös
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引用次数: 10
Recent progress in cannabinoid research. 大麻素研究的最新进展。
Q1 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2006-01-01 DOI: 10.1016/S0079-6468(05)44406-9
Julia Adam, Phillip M Cowley, Takao Kiyoi, Angus J Morrison, Christopher J W Mort
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引用次数: 7
Peptide deformylase inhibitors. 肽去甲酰基酶抑制剂。
Q1 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2006-01-01 DOI: 10.1016/S0079-6468(05)44403-3
Kelly Aubart, Magdalena Zalacain
{"title":"Peptide deformylase inhibitors.","authors":"Kelly Aubart, Magdalena Zalacain","doi":"10.1016/S0079-6468(05)44403-3","DOIUrl":"https://doi.org/10.1016/S0079-6468(05)44403-3","url":null,"abstract":"","PeriodicalId":20755,"journal":{"name":"Progress in medicinal chemistry","volume":null,"pages":null},"PeriodicalIF":0.0,"publicationDate":"2006-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/S0079-6468(05)44403-3","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"26023347","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
期刊
Progress in medicinal chemistry
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