Pub Date : 2013-01-01DOI: 10.1016/B978-0-444-62652-3.10000-6
Geoff Lawton, David R Witty
{"title":"Glucokinase. Preface.","authors":"Geoff Lawton, David R Witty","doi":"10.1016/B978-0-444-62652-3.10000-6","DOIUrl":"https://doi.org/10.1016/B978-0-444-62652-3.10000-6","url":null,"abstract":"","PeriodicalId":20755,"journal":{"name":"Progress in medicinal chemistry","volume":"52 ","pages":"v-vii"},"PeriodicalIF":0.0,"publicationDate":"2013-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/B978-0-444-62652-3.10000-6","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"31217739","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
Pub Date : 2013-01-01DOI: 10.1016/B978-0-444-62652-3.00003-X
Félix Calderón, David M Wilson, Francisco-Javier Gamo
{"title":"Antimalarial drug discovery: recent progress and future directions.","authors":"Félix Calderón, David M Wilson, Francisco-Javier Gamo","doi":"10.1016/B978-0-444-62652-3.00003-X","DOIUrl":"https://doi.org/10.1016/B978-0-444-62652-3.00003-X","url":null,"abstract":"","PeriodicalId":20755,"journal":{"name":"Progress in medicinal chemistry","volume":"52 ","pages":"97-151"},"PeriodicalIF":0.0,"publicationDate":"2013-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/B978-0-444-62652-3.00003-X","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"31217737","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
Pub Date : 2013-01-01DOI: 10.1016/B978-0-444-62652-3.00002-8
Lyn H Jones, David A Price
{"title":"Medicinal chemistry of glucagon-like peptide receptor agonists.","authors":"Lyn H Jones, David A Price","doi":"10.1016/B978-0-444-62652-3.00002-8","DOIUrl":"https://doi.org/10.1016/B978-0-444-62652-3.00002-8","url":null,"abstract":"","PeriodicalId":20755,"journal":{"name":"Progress in medicinal chemistry","volume":"52 ","pages":"45-96"},"PeriodicalIF":0.0,"publicationDate":"2013-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/B978-0-444-62652-3.00002-8","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"31217736","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
Pub Date : 2013-01-01DOI: 10.1016/B978-0-444-62652-3.00001-6
Darren McKerrecher, Michael J Waring
{"title":"Property-based design in the optimisation of benzamide glucokinase activators: from hit to clinic.","authors":"Darren McKerrecher, Michael J Waring","doi":"10.1016/B978-0-444-62652-3.00001-6","DOIUrl":"https://doi.org/10.1016/B978-0-444-62652-3.00001-6","url":null,"abstract":"","PeriodicalId":20755,"journal":{"name":"Progress in medicinal chemistry","volume":"52 ","pages":"1-43"},"PeriodicalIF":0.0,"publicationDate":"2013-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/B978-0-444-62652-3.00001-6","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"31217735","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
Pub Date : 2012-01-01DOI: 10.1016/B978-0-12-396493-9.00002-9
Michael E Kort, Philip R Kym
{"title":"TRPV1 antagonists: clinical setbacks and prospects for future development.","authors":"Michael E Kort, Philip R Kym","doi":"10.1016/B978-0-12-396493-9.00002-9","DOIUrl":"https://doi.org/10.1016/B978-0-12-396493-9.00002-9","url":null,"abstract":"","PeriodicalId":20755,"journal":{"name":"Progress in medicinal chemistry","volume":"51 ","pages":"57-70"},"PeriodicalIF":0.0,"publicationDate":"2012-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/B978-0-12-396493-9.00002-9","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"40171223","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
Pub Date : 2012-01-01DOI: 10.1016/B978-0-12-396493-9.00003-0
Adam D Hughes, Alexander McNamara, Tod Steinfeld
{"title":"Multivalent dual pharmacology muscarinic antagonist and β₂ agonist (MABA) molecules for the treatment of COPD.","authors":"Adam D Hughes, Alexander McNamara, Tod Steinfeld","doi":"10.1016/B978-0-12-396493-9.00003-0","DOIUrl":"https://doi.org/10.1016/B978-0-12-396493-9.00003-0","url":null,"abstract":"","PeriodicalId":20755,"journal":{"name":"Progress in medicinal chemistry","volume":"51 ","pages":"71-95"},"PeriodicalIF":0.0,"publicationDate":"2012-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/B978-0-12-396493-9.00003-0","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"40171224","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
Pub Date : 2012-01-01DOI: 10.1016/B978-0-12-396493-9.00005-4
G Lawton, David R Witty
{"title":"The large scale restructuring of pharmaceutical company research function. Preface.","authors":"G Lawton, David R Witty","doi":"10.1016/B978-0-12-396493-9.00005-4","DOIUrl":"https://doi.org/10.1016/B978-0-12-396493-9.00005-4","url":null,"abstract":"","PeriodicalId":20755,"journal":{"name":"Progress in medicinal chemistry","volume":"51 ","pages":"v-vi"},"PeriodicalIF":0.0,"publicationDate":"2012-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/B978-0-12-396493-9.00005-4","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"40171226","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
Pub Date : 2011-01-01DOI: 10.1016/B978-0-12-381290-2.00001-X
Graham F Smith
{"title":"Designing drugs to avoid toxicity.","authors":"Graham F Smith","doi":"10.1016/B978-0-12-381290-2.00001-X","DOIUrl":"https://doi.org/10.1016/B978-0-12-381290-2.00001-X","url":null,"abstract":"","PeriodicalId":20755,"journal":{"name":"Progress in medicinal chemistry","volume":"50 ","pages":"1-47"},"PeriodicalIF":0.0,"publicationDate":"2011-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/B978-0-12-381290-2.00001-X","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"29667943","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}