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Quasicrystals at high pressures and temperatures: a review 高压和高温下的准晶体:综述
IF 2 4区 综合性期刊 Q2 MULTIDISCIPLINARY SCIENCES Pub Date : 2023-08-04 DOI: 10.1007/s12210-023-01183-z
V. Stagno, L. Bindi
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引用次数: 0
Detailed dynamics of bimolecular recombination of heavy atomic ions 重原子离子双分子复合的详细动力学
IF 2 4区 综合性期刊 Q2 MULTIDISCIPLINARY SCIENCES Pub Date : 2023-08-04 DOI: 10.1007/s12210-023-01182-0
V. Akimov, V. M. Azriel, E. V. Ermolova, D. B. Kabanov, L. I. Kolesnikova, L. Rusin, M. Sevryuk
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引用次数: 0
Vegetation composition and structure of Dabena woodland in western Ethiopia 埃塞俄比亚西部达比纳林地植被组成与结构
IF 2 4区 综合性期刊 Q2 MULTIDISCIPLINARY SCIENCES Pub Date : 2023-08-03 DOI: 10.1007/s12210-023-01181-1
Kifle Yeshitila, T. Bekele, T. Wondimu, S. Demissew
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引用次数: 0
Prediction of solar cycle 25: applications and comparison 太阳活动周期25的预测:应用与比较
IF 2 4区 综合性期刊 Q2 MULTIDISCIPLINARY SCIENCES Pub Date : 2023-07-29 DOI: 10.1007/s12210-023-01184-y
V. Penza, L. Bertello, Matteo Cantoresi, S. Criscuoli, F. Berrilli
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引用次数: 0
Utilization of agro-industrial biowastes to produce xylanase using Aspergillus niger AUMC 14230: optimization of production parameters 利用黑曲霉AUMC 14230生产木聚糖酶农工废弃物:生产参数的优化
IF 2 4区 综合性期刊 Q2 MULTIDISCIPLINARY SCIENCES Pub Date : 2023-07-26 DOI: 10.1007/s12210-023-01180-2
Y. F. Abdelaliem, Marwa Hamdy Mahmoud, Nabil Abo Elkassem, S. Mansour, M. Ramadan, A. Mohdaly
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引用次数: 0
Mathematical aspects of quasicrystals 准晶体的数学方面
IF 2 4区 综合性期刊 Q2 MULTIDISCIPLINARY SCIENCES Pub Date : 2023-07-26 DOI: 10.1007/s12210-023-01176-y
C. Sbordone, M. Guida
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引用次数: 0
The flax in the “Flora’s image” in the Ariadne House (Pompeian area, Italy) as a symbol of feminine in a wedding sacred to the afterlife 在阿里阿德涅宫(意大利庞贝地区)的“弗洛拉的形象”中,亚麻是来世神圣婚礼中女性的象征
IF 2 4区 综合性期刊 Q2 MULTIDISCIPLINARY SCIENCES Pub Date : 2023-07-18 DOI: 10.1007/s12210-023-01177-x
G. Caneva, A. Bourmaud, A. Bellini, A. Melelli
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引用次数: 1
The kombucha ingestion benefits on the intestinal microbiota 康普茶对肠道菌群有益
IF 2 4区 综合性期刊 Q2 MULTIDISCIPLINARY SCIENCES Pub Date : 2023-07-18 DOI: 10.1007/s12210-023-01178-w
Iraíldo Francisco Soares, Michele Alves de Lima, M. Lucarini, A. Durazzo, D. Arcanjo, Simone Kelly Rodrigues Lima, R. D. da Silva
{"title":"The kombucha ingestion benefits on the intestinal microbiota","authors":"Iraíldo Francisco Soares, Michele Alves de Lima, M. Lucarini, A. Durazzo, D. Arcanjo, Simone Kelly Rodrigues Lima, R. D. da Silva","doi":"10.1007/s12210-023-01178-w","DOIUrl":"https://doi.org/10.1007/s12210-023-01178-w","url":null,"abstract":"","PeriodicalId":54501,"journal":{"name":"Rendiconti Lincei-Scienze Fisiche E Naturali","volume":"66 1","pages":"833 - 841"},"PeriodicalIF":2.0,"publicationDate":"2023-07-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"78393874","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"综合性期刊","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Soil quality assessment based on MCDA–GIS hybrid approach for sustainable hazelnut farming under humid ecosystem environment 湿润生态环境下基于MCDA-GIS的榛子可持续种植土壤质量评价
IF 2 4区 综合性期刊 Q2 MULTIDISCIPLINARY SCIENCES Pub Date : 2023-07-18 DOI: 10.1007/s12210-023-01179-9
B. Bayraklı, O. Dengiz, N. Kars
{"title":"Soil quality assessment based on MCDA–GIS hybrid approach for sustainable hazelnut farming under humid ecosystem environment","authors":"B. Bayraklı, O. Dengiz, N. Kars","doi":"10.1007/s12210-023-01179-9","DOIUrl":"https://doi.org/10.1007/s12210-023-01179-9","url":null,"abstract":"","PeriodicalId":54501,"journal":{"name":"Rendiconti Lincei-Scienze Fisiche E Naturali","volume":"17 1","pages":"921 - 940"},"PeriodicalIF":2.0,"publicationDate":"2023-07-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"82576975","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"综合性期刊","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 1
Old tricks and new trends to address tumors: a medicinal chemist’s perspective 治疗肿瘤的老方法和新趋势:一个药物化学家的观点
IF 2 4区 综合性期刊 Q2 MULTIDISCIPLINARY SCIENCES Pub Date : 2023-07-13 DOI: 10.4081/scienze.2022.826
P. Seneci
Major efforts in the past decades have provided novel small molecule drugs and biologicals and innovative mechanisms against tumors, but the quest for safer, bioavailable and more effective active principles is still ongoing. This contribution focuses on innovative approaches to fulfill therapeutic goals in oncology; namely, the inhibition of the stabilizing interaction between the RNA-binding protein HuR and mRNAs of multiple oncogenes, and the unleashing of a strong immune reaction against cancer cells by antagonizing the PD-1 – PD-L1 interaction on the surface of cancer cells. “Classical” drug-like, bioavailable small molecules were either rationally designed from a naturally occurring template (tanshinones converted to aza-tanshinones – HuR), or from a synthetic peptidomimetic inhibitor (biphenyloxy aryls converted to disubstituted triazines – PD-L1); after their synthesis and activity profiling, early leads were identified to be further structurally optimized in the near future.
在过去的几十年里,主要的努力已经提供了新的小分子药物和生物制剂以及抗肿瘤的创新机制,但对更安全、生物可利用性和更有效的活性原理的追求仍在进行中。该贡献侧重于实现肿瘤学治疗目标的创新方法;即抑制rna结合蛋白HuR与多种癌基因mrna之间的稳定相互作用,通过拮抗癌细胞表面的PD-1 - PD-L1相互作用,对癌细胞产生强烈的免疫反应。“经典”类药物,生物可利用的小分子要么从自然存在的模板(丹参酮转化为aza-丹参酮- HuR)合理设计,要么从合成的拟肽抑制剂(联苯氧基芳基转化为二取代三嗪- PD-L1)设计;在对其进行合成和活性分析后,确定了早期先导物,并在不久的将来进行进一步的结构优化。
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引用次数: 0
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