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Drug Metabolism and Pharmacokinetics最新文献

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Drug metabolism: A half-century plus of progress, continued needs, and new opportunities 药物代谢:半个多世纪的进步、持续需求和新机遇
IF 2.1 4区 医学 Q2 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2024-04-01 DOI: 10.1016/j.dmpk.2023.100561
F. Peter Guengerich
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引用次数: 0
Identification and characterization of novel metabolites of F2-isoprostanes F2- 异前列腺素新型代谢物的鉴定和表征
IF 2.1 4区 医学 Q2 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2024-04-01 DOI: 10.1016/j.dmpk.2023.100806
Marina Nogueira , Stephanie Sanchez , Benlian Gao , Warda Amin , Sarah Thomas , Gong Yang , Ginger Milne
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引用次数: 0
Projections for future challenges and opportunities for pharmacokineticists 对药物动力学家未来挑战和机遇的预测
IF 2.1 4区 医学 Q2 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2024-04-01 DOI: 10.1016/j.dmpk.2023.100597
Joseph Balthasar
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引用次数: 0
Potential ADME-related issues for PROTACs PROTAC 的潜在 ADME 相关问题
IF 2.1 4区 医学 Q2 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2024-04-01 DOI: 10.1016/j.dmpk.2023.100590
Matthew Hoffman
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引用次数: 0
Successful optimization of pharmacokinetics and pharmacodynamics of oral cyclic peptide PCSK9 inhibitors 成功优化口服环肽 PCSK9 抑制剂的药代动力学和药效学
IF 2.1 4区 医学 Q2 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2024-04-01 DOI: 10.1016/j.dmpk.2023.100591
Tjerk JH. Bueters
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引用次数: 0
Microbiome impacts on drug metabolism 微生物组对药物代谢的影响
IF 2.1 4区 医学 Q2 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2024-04-01 DOI: 10.1016/j.dmpk.2023.100592
Andrew Goodman
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引用次数: 0
Smart compound library based on machine learning, sensing technology, and programmable logic control 基于机器学习、传感技术和可编程逻辑控制的智能化合物库
IF 2.1 4区 医学 Q2 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2024-04-01 DOI: 10.1016/j.dmpk.2023.100824
Hongye Li, Minhao Fang, Xiangling Wang, Jindi Shi, Wei Zhao, Yi Tao, Liang Shen
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引用次数: 0
Mathematical modeling of affinity design goals for CIS-binding BI-specific antibody-based molecules 基于 CIS 结合 BI 特异性抗体分子的亲和力设计目标的数学建模
IF 2.1 4区 医学 Q2 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2024-04-01 DOI: 10.1016/j.dmpk.2023.100577
Isabel Figueroa
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引用次数: 0
Development of a simple, fast inhibition assay for rat CYP3A enzymes 为大鼠 CYP3A 酶开发一种简单、快速的抑制测定法
IF 2.1 4区 医学 Q2 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2024-04-01 DOI: 10.1016/j.dmpk.2023.100834
Michael Voice, Andrew Shepherd, Gillian Dixon
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引用次数: 0
Strategies for de-risking n-nitrosamine impurities in APIS 消除 APIS 中正亚硝胺杂质风险的策略
IF 2.1 4区 医学 Q2 Pharmacology, Toxicology and Pharmaceutics Pub Date : 2024-04-01 DOI: 10.1016/j.dmpk.2023.100581
Joel Bercu
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引用次数: 0
期刊
Drug Metabolism and Pharmacokinetics
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