Pub Date : 2024-05-13DOI: 10.1016/j.dmpk.2023.100898
Tingting Yan, Nana Yan, Yangliu Xia, Haiping Hao, Frank J. Gonzalez
{"title":"Hepatocyte CEBPA restricts the progression of liver fibrosis","authors":"Tingting Yan, Nana Yan, Yangliu Xia, Haiping Hao, Frank J. Gonzalez","doi":"10.1016/j.dmpk.2023.100898","DOIUrl":"https://doi.org/10.1016/j.dmpk.2023.100898","url":null,"abstract":"","PeriodicalId":11298,"journal":{"name":"Drug Metabolism and Pharmacokinetics","volume":null,"pages":null},"PeriodicalIF":2.1,"publicationDate":"2024-05-13","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"141518089","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"医学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
Pub Date : 2024-05-13DOI: 10.1016/j.dmpk.2023.100990
Acilegna Rodriguez, Megan Graves, Yewei Du, Roberta Kaufman, Jian-Lu Chen, Makenzie Sacca, Mark Warren
{"title":"Monocarboxylate transporter 10: substrate-dependent mode of transport","authors":"Acilegna Rodriguez, Megan Graves, Yewei Du, Roberta Kaufman, Jian-Lu Chen, Makenzie Sacca, Mark Warren","doi":"10.1016/j.dmpk.2023.100990","DOIUrl":"https://doi.org/10.1016/j.dmpk.2023.100990","url":null,"abstract":"","PeriodicalId":11298,"journal":{"name":"Drug Metabolism and Pharmacokinetics","volume":null,"pages":null},"PeriodicalIF":2.1,"publicationDate":"2024-05-13","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"141058807","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"医学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Substrate-dependent characteristics in the transport function of SLC19A3: examination of the aspect of its sensitivity to flavonoids","authors":"Hiroaki Yuasa, Saena Yamashita, Takahiro Yamashiro, Tomoya Yasujima","doi":"10.1016/j.dmpk.2023.100993","DOIUrl":"https://doi.org/10.1016/j.dmpk.2023.100993","url":null,"abstract":"","PeriodicalId":11298,"journal":{"name":"Drug Metabolism and Pharmacokinetics","volume":null,"pages":null},"PeriodicalIF":2.1,"publicationDate":"2024-05-13","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"141058823","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"医学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
Pub Date : 2024-05-13DOI: 10.1016/j.dmpk.2023.100959
Kyungsun Moon, Sung-Hoon Ahn
{"title":"Pharmacokinetics of perfluoroocanoic acid and perfluorohexane sulfonic acid in various rat models","authors":"Kyungsun Moon, Sung-Hoon Ahn","doi":"10.1016/j.dmpk.2023.100959","DOIUrl":"https://doi.org/10.1016/j.dmpk.2023.100959","url":null,"abstract":"","PeriodicalId":11298,"journal":{"name":"Drug Metabolism and Pharmacokinetics","volume":null,"pages":null},"PeriodicalIF":2.1,"publicationDate":"2024-05-13","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"141058987","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"医学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
Pub Date : 2024-05-13DOI: 10.1016/j.dmpk.2023.100943
Iain Shaw, Adam Robinson-Miller, Phil Evans, Stuart Mair
{"title":"The practical impact of the FDA draft guidance on human mass balance studies – a year of client discussions","authors":"Iain Shaw, Adam Robinson-Miller, Phil Evans, Stuart Mair","doi":"10.1016/j.dmpk.2023.100943","DOIUrl":"https://doi.org/10.1016/j.dmpk.2023.100943","url":null,"abstract":"","PeriodicalId":11298,"journal":{"name":"Drug Metabolism and Pharmacokinetics","volume":null,"pages":null},"PeriodicalIF":2.1,"publicationDate":"2024-05-13","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"141058991","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"医学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Encequidar is a gut-restricted P-GP specific inhibitor that boosts oral bioavailability and inhibits intestinal secretion in rats and dogs.","authors":"Murali Subramanian, Aaliyah Shodeinde, Gregg Schwarzwalder, Ana Gonzalez, Josh Yu, Guangyu Zhao, Jia Hao, Xiaomin Liang, Yurong Lai, Raju Subramanian","doi":"10.1016/j.dmpk.2023.100989","DOIUrl":"https://doi.org/10.1016/j.dmpk.2023.100989","url":null,"abstract":"","PeriodicalId":11298,"journal":{"name":"Drug Metabolism and Pharmacokinetics","volume":null,"pages":null},"PeriodicalIF":2.1,"publicationDate":"2024-05-13","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"141058821","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"医学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
Pub Date : 2024-05-13DOI: 10.1016/j.dmpk.2023.100933
Ping Lu, Randy Miller, Jianmei Pang, Sheri Smith, Jason Hoar, Mark Concilla
{"title":"In vivo and in vitro biotransformation of molnupiravir (MOV), An oral prodrug of the antiviral ribonucleoside analog Β-D-N4-hydroxycytidine (NHC)","authors":"Ping Lu, Randy Miller, Jianmei Pang, Sheri Smith, Jason Hoar, Mark Concilla","doi":"10.1016/j.dmpk.2023.100933","DOIUrl":"https://doi.org/10.1016/j.dmpk.2023.100933","url":null,"abstract":"","PeriodicalId":11298,"journal":{"name":"Drug Metabolism and Pharmacokinetics","volume":null,"pages":null},"PeriodicalIF":2.1,"publicationDate":"2024-05-13","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"141058860","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"医学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}